Agent Pharmacokinetic parameters(unit) Geometric Mean Geometric Mean Ratios (90% CI) CV (%)
Famitinib + Omeprazole Famitinib
Famitinib Cmax (ng/mL) 42.0 42.5 0.989(0.953, 1.027) 6.8
AUC0-t (h·ng/mL) 1333.2 1395.0 0.956(0.907, 1.007) 9.5
AUC0-∞ (h·ng/mL) 1351.9 1417.9 0.953(0.905, 1.005) 9.6
SHR116637 Cmax (ng/mL) 1.5 1.9 0.851(0.786, 0.920) 14.5
AUC0-t (h·ng/mL) 96.3 108.2 0.890(0.838, 0.946) 11.1
AUC0-∞ (h·ng/mL) 105.5 118.9 0.887(0.835, 0.943) 11.2